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Search Results for " histone acetyltransferase "

20

Compounds

Cat No. Product Name Synonyms Targets
T11563 Histone Acetyltransferase Inhibitor II Epigenetic Reader Domain , Histone Acetyltransferase
Histone Acetyltransferase Inhibitor II is a selective and cell permeable inhibitor of p300 histone acetyltransferase(IC50 : 5 μM).with anti-acetylase activity in mammalian cells.
T77560 Histone acetyltransferase p300 Inhibitor 4c Carbonic Anhydrase , AChE
Histone acetyltransferase p300 Inhibitor 4c is a 2-aminothiazole derivative. Histone acetyltransferase p300 Inhibitor 4c inhibited hCA I, hCA II, AChE and BChE with Ki values of 0.008 ± 0.001, 0.124 ± 0.017, 0.129 ± 0.03...
T3499 Remodelin Histone Acetyltransferase
Remodelin is an effective and specific inhibitor of the acetyl-transferase protein NAT10.
T8344 CPTH2 Apoptosis , Histone Acetyltransferase
CPTH2 is a histone acetyltransferase inhibitor modulating Gcn5 network.
T12098 MOZ-IN-2 Histone Acetyltransferase
MOZ-IN-2 is an protein MOZ inhibitor(IC50 of 125 μM).
T11807 L002 Others , Histone Acetyltransferase , STAT
L002, a potent, cell-permeable, reversible, and specific acetyltransferase p300 (KAT3B) inhibitor with an IC50 of 1.98 μM, directly binds the acetyl-CoA pocket and competitively inhibits the FATp300 catalytic domain. By ...
T6133 Remodelin hydrobromide Remodelin,Remodelin HBR RAAS , Histone Acetyltransferase
Remodelin hydrobromide (Remodelin HBR) is a novel potent and selective inhibitor of the acetyl-transferase protein NAT10.
T5468 YF-2 Others , Epigenetic Reader Domain , Histone Acetyltransferase
YF-2 is blood-brain-barrier permeable histone acetyltransferase activator, acetylates H3 in the hippocampus, CBP, PCAF, and GCN5 with EC50s of 2.75 μM, 29.04 μM and 49.31 μM , respectively
T4679 WM-1119 WM1119 Histone Acetyltransferase
WM-1119 is a highly potent, selective KAT6A/B inhibitor
T15216 EML 425 Epigenetic Reader Domain , Histone Acetyltransferase
EML 425 is a potent and selective inhibitor of CREB binding protein (CBP)/p300 (IC50s: 2.9 and 1.1 μM, respectively).
T15405 GNE-781 Epigenetic Reader Domain
GNE-781 is a highly potent and selective inhibitor of CBP (IC50: 0.94 nM in TR-FRET assay). GNE-781 also inhibits BRET and BRD4(1) (IC50s: 6.2 nM and 5100 nM, respectively).
T14073 A-485 Epigenetic Reader Domain , Histone Acetyltransferase
A-485 is a potent and selective catalytic p300/CBP inhibitor(IC50s of 9.8 nM and 2.6 nM for p300 and CBP, respectively).
T2452 C646 Apoptosis , Epigenetic Reader Domain , Histone Acetyltransferase , Autophagy
C646, a histone acetyltransferase inhibitor, inhibits p300 (Ki: 400 nM, in a cell-free assay).
T8778 TTK21 Epigenetic Reader Domain
TTK21 is an activator of CBP/p300 histone acetyltransferase activity.
T6811 CPI-637 CPI 637 Epigenetic Reader Domain , Histone Acetyltransferase
CPI-637 is a selective and cell-active benzodiazepinone CBP/EP300 bromodomain inhibitor.
T11366 Garcinol Apoptosis , Endogenous Metabolite , Histone Acetyltransferase , AChR , AChE
Garcinol also inhibits histone acetyltransferases (HATs, IC50= 7 μM) and p300/CPB-associated factor (PCAF, IC50 = 5 μM). Garcinol has anti-inflammatory and anti-cancer activity. Garcinol, a polyisoprenylated benzophenone...
T3969 I-CBP112 Epigenetic Reader Domain , Histone Acetyltransferase
I-CBP112 is a specific and potent acetyl-lysine competitive protein-protein interaction inhibitor targeting the CBP/p300 bromodomains.
T9541 CTB Cholera Toxin B subunit Epigenetic Reader Domain
CTB (Cholera Toxin B subunit) is an activator of p300 histone acetyltransferase and induces apoptosis in MCF-7 cells.
T4362 WM-8014 MOZ-IN-3 Histone Acetyltransferase
WM-8014 (MOZ-IN-3) is an inhibitor of MOZ(IC50=55 nM), a member of histone acetyltransferases.
TN1150 Procyanidin B3 Histone Acetyltransferase
Procyanidin B3(B3) is a procyanidin dimer that is widely studied due to its high abundance in the human diet and antioxidant activity.

Compounds

Histone Acetyltransferase Inhibitor II
T11563
Synonym:
Target: Epigenetic Reader Domain, Histone Acetyltransferase
Histone acetyltransferase p300 Inhibitor 4c
T77560
Synonym:
Target: Carbonic Anhydrase, AChE
Remodelin
T3499
Synonym:
Target: Histone Acetyltransferase
CPTH2
T8344
Synonym:
Target: Apoptosis, Histone Acetyltransferase
MOZ-IN-2
T12098
Synonym:
Target: Histone Acetyltransferase
L002
T11807
Synonym:
Target: Others, Histone Acetyltransferase, STAT
Remodelin hydrobromide
T6133
Synonym: Remodelin,Remodelin HBR
Target: RAAS, Histone Acetyltransferase
YF-2
T5468
Synonym:
Target: Others, Epigenetic Reader Domain, Histone Acetyltransferase
WM-1119
T4679
Synonym: WM1119
Target: Histone Acetyltransferase
EML 425
T15216
Synonym:
Target: Epigenetic Reader Domain, Histone Acetyltransferase
GNE-781
T15405
Synonym:
Target: Epigenetic Reader Domain
A-485
T14073
Synonym:
Target: Epigenetic Reader Domain, Histone Acetyltransferase
C646
T2452
Synonym:
Target: Apoptosis, Epigenetic Reader Domain, Histone Acetyltransferase, Autophagy
TTK21
T8778
Synonym:
Target: Epigenetic Reader Domain
CPI-637
T6811
Synonym: CPI 637
Target: Epigenetic Reader Domain, Histone Acetyltransferase
Garcinol
T11366
Synonym:
Target: Apoptosis, Endogenous Metabolite, Histone Acetyltransferase, AChR, AChE
I-CBP112
T3969
Synonym:
Target: Epigenetic Reader Domain, Histone Acetyltransferase
CTB
T9541
Synonym: Cholera Toxin B subunit
Target: Epigenetic Reader Domain
WM-8014
T4362
Synonym: MOZ-IN-3
Target: Histone Acetyltransferase
Procyanidin B3
TN1150
Synonym:
Target: Histone Acetyltransferase
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TargetMol